RNA-UNY 2010 program

SOMAmers: Proteomics to lung cancer to a Wellness Chip

Larry Gold

University of Colorado at Boulder and SomaLogic, Inc.

We figured out a way to make novel aptamers, called SOMAmers. The SOMAmers, made of modified single-stranded DNA, have high affinities for their target human proteins, and in addition have very slow off-rates. The high binding quality of these special aptamers is supported by a crystal structure of one such SOMAmer with its protein partner.

We also figured out a way to use the SOMAmers to do deep proteomics. Today we measure 1,100 human proteins in serum, plasma, or tissue extracts, using only 15 µl of sample. The measurements are accurate (CVs of ~ 5%) and very sensitive; more than half the proteins are measured with limits of detection below pM. The combination of reagents and a novel assay has made biomarker discovery relatively easy. And thats what we do ...

We get samples from healthy and sick people and do an unbiased experiment by asking if any proteins on the menu go up or down in the blood of sick people. We have found many blood biomarkers for lung cancer, mesothelioma, pancreatic cancer, and more.

Lung cancer is the leading cause of cancer deaths. Most cases are diagnosed at an advanced stage. Patients diagnosed at an early stage who have surgery experience an 86% overall 5-year survival thus one needs earlier detection of lung cancer.

I will share data from a large clinical trial (almost 1,400 subjects) from four independent studies of long-term tobacco-exposed populations. We identified 44 candidate biomarkers, from which a 12- protein panel was constructed. The panel identified NSCLC from controls with 91% sensitivity and 84% specificity in the training set, and 89% sensitivity and 83% specificity in the blinded, independent verification set. Performance was similar for early and late stage disease.

We also have compared protein concentrations in NSCLC biopsy materials with literature values for mRNA concentrations in similar biopsies. The correlations between proteins and their mRNAs are poor, suggesting that a discovery proteomics platform might be essential for understanding NSCLC biology.

Finally, with only some trepidation, I will describe our goal of transforming medicine through a Wellness Chip, aimed at the most devastating diseases for which early diagnosis and action could be life-saving.

RNA-UNY 2010 program